Affinity DataKi: 1nMAssay Description:Evaluated for the Non competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Inhibition of HDAC in human HeLa cell lysates after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 215nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 249nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 2.52E+3nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 8.06E+3nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 1.16E+4nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of CDK4/Cyclin D1 complex formationMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of CDK4/Cyclin D1 complex formationMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+5nMpH: 6.0Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
Affinity DataKd: 5.90E+5nMpH: 7.5Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
Affinity DataKd: 5.30E+5nMpH: 7.5Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at GAL4-fused human PPARalpha LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.60E+3nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.60E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.83E+4nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 0.280nMAssay Description:Agonist activity at GAL4-fused human PPARgamma LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.50E+4nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in reporter combo cells after 36 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 5.24E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.53E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 8.90E+3nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 83nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair