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Found 99 from University of Oklahoma
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031347(2-Amino-5-(2-amino-propyl)-benzene-1,4-diol | CHEM...)
Affinity DataKi:  1nMAssay Description:Evaluated for the Non competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031347(2-Amino-5-(2-amino-propyl)-benzene-1,4-diol | CHEM...)
Affinity DataKi:  3nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031343(2-Amino-5-(2-amino-ethyl)-benzene-1,4-diol | CHEMB...)
Affinity DataKi:  5nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031341(4-Amino-5-(2-amino-propyl)-benzene-1,2-diol | CHEM...)
Affinity DataKi:  8nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031343(2-Amino-5-(2-amino-ethyl)-benzene-1,4-diol | CHEMB...)
Affinity DataKi:  9nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031341(4-Amino-5-(2-amino-propyl)-benzene-1,2-diol | CHEM...)
Affinity DataKi:  9nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031344(4-Amino-5-(2-amino-ethyl)-benzene-1,2-diol | CHEMB...)
Affinity DataKi:  11nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM81264(5-(2-aminoethyl)benzene-1,2,4-triol;hydrobromide |...)
Affinity DataKi:  12nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031346(4-Amino-6-(2-amino-ethyl)-benzene-1,3-diol | CHEMB...)
Affinity DataKi:  13nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031342(5-(2-Amino-propyl)-benzene-1,2,4-triol | 5-(2-Amin...)
Affinity DataKi:  16nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031344(4-Amino-5-(2-amino-ethyl)-benzene-1,2-diol | CHEMB...)
Affinity DataKi:  17nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031342(5-(2-Amino-propyl)-benzene-1,2,4-triol | 5-(2-Amin...)
Affinity DataKi:  26nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031348(4-Amino-6-(2-amino-propyl)-benzene-1,3-diol | CHEM...)
Affinity DataKi:  46nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031346(4-Amino-6-(2-amino-ethyl)-benzene-1,3-diol | CHEMB...)
Affinity DataKi:  47nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM81264(5-(2-aminoethyl)benzene-1,2,4-triol;hydrobromide |...)
Affinity DataKi:  51nMAssay Description:Evaluated for the Competitive inhibition of uptake of norepinephrineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50031348(4-Amino-6-(2-amino-propyl)-benzene-1,3-diol | CHEM...)
Affinity DataKi:  112nMAssay Description:Evaluated for the Competitive inhibition of uptake of dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50049427(CHEMBL3315350)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of HDAC in human HeLa cell lysates after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50451132(CHEMBL2079586 | WIN-35428)
Affinity DataIC50:  24nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50454604(CHEMBL2112302)
Affinity DataIC50:  25nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50454606(CHEMBL2112303)
Affinity DataIC50:  70nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50454605(CHEMBL2112304)
Affinity DataIC50:  153nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50454607(CHEMBL2112300)
Affinity DataIC50:  215nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  249nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50454609(CHEMBL2112305)
Affinity DataIC50:  1.18E+3nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50454608(CHEMBL2112306)
Affinity DataIC50:  2.52E+3nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50059315((S)-4-(4-Iodo-benzoyloxy)-1-methyl-piperidine-3-ca...)
Affinity DataIC50:  8.06E+3nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50059308(4-Iodo-benzoic acid 1-methyl-piperidin-4-yl ester ...)
Affinity DataIC50:  1.16E+4nMAssay Description:Compound was tested for inhibitory activity to displace [3H]WIN-35428 at dopamine transporter in Rat Striatal Membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50478536(Halistanol Sulfate)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of CDK4/Cyclin D1 complex formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50478545(Siphonodictyal C)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of CDK4/Cyclin D1 complex formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEfflux pump membrane transporter(Escherichia coli)
University of Oklahoma

LigandPNGBDBM81507(MC-207,110)
Affinity DataKd:  1.10E+5nMpH: 6.0Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEfflux pump membrane transporter(Escherichia coli)
University of Oklahoma

LigandPNGBDBM81507(MC-207,110)
Affinity DataKd:  5.90E+5nMpH: 7.5Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEfflux pump membrane transporter(Escherichia coli)
University of Oklahoma

LigandPNGBDBM282((3R,4S,5R,6R)-5-hydroxy-6-[(2-hydroxy-3-{[4-hydrox...)
Affinity DataKd:  5.30E+5nMpH: 7.5Assay Description:Binding of inhibitors and substrates to immobilized AcrB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50013727(CHEBI:79990 | CHEMBL410478 | GW409544)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at GAL4-fused human PPARalpha LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  1.83E+4nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50013727(CHEBI:79990 | CHEMBL410478 | GW409544)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at GAL4-fused human PPARgamma LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462441(CHEMBL1565327)
Affinity DataEC50:  2.50E+4nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in reporter combo cells after 36 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462441(CHEMBL1565327)
Affinity DataEC50:  5.24E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  2.53E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  8.90E+3nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
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